SCHEMBL10754174

SCHEMBL10754174

NS(=O)(=O)c1ccc(-c2cn3ncccc3n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 18/20 0.51
CA1 P00915 17/20 0.51
CA12 O43570 17/20 0.51
CA9 Q16790 17/20 0.51
CA7 P43166 1/20 0.46
HDAC6 Q9UBN7 1/20 0.45
CA5A P35218 2/20 0.44
CA5B Q9Y2D0 2/20 0.44
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
GFER P55789 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
PTGS2 P35354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10752677 0.82 ALDH1A1 (0.64) HDAC6KDM4ENPC1ALDH1A1HPGD
SCHEMBL10756399 0.80 RAB9A (0.46) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL10758245 0.79 HDAC6 (0.42) HDAC6KDM4ENPC1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL10758246 0.78 HDAC6 (0.41) HDAC6KDM4ENPC1ALDH1A1HPGD
SCHEMBL1202800 0.77 ALDH1A1 (0.49) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL10754655 0.77 HDAC6 (0.74) HDAC6KDM4ENPC1ALDH1A1HPGD
SCHEMBL12970200 0.76 RAB9A (0.55) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL5309811 0.76 NPC1 (0.57) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL15473569 0.76 NPC1 (0.57) KDM4ENPC1ALDH1A1RAB9A
SCHEMBL10755848 0.76 KLK7 (0.56) HDAC6KDM4ENPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4716169-A INOTROPIC AGENTS DR. KARL THOMAE GMBH (DE) 1987-12-29 US disclosed
EP-0185345-A1 Imidazo derivatives, their preparation and medicines containing them Dr. Karl Thomae GmbH (DE) 1986-06-25 EP disclosed