SCHEMBL10757294

SCHEMBL10757294

COc1ccsc1C1OC(=O)NC1=O

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.52
KEAP1 Q14145 1/20 0.33
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10760577 0.80 CA2 (0.46) CA2KDM4ECYP1A2CYP3A4GAA
SCHEMBL10759314 0.76 CA2 (0.46) CA2
SCHEMBL10763085 0.76 CA2 (0.46) CA2
SCHEMBL11043589 0.72 CA2 (0.67) CA2KDM4EMAPTMEN1KMT2A
SCHEMBL10757512 0.72 CA2 (0.48) CA2
SCHEMBL10759946 0.71 CA2 (0.57) CA2
SCHEMBL10759552 0.71 CA2 (0.54) CA2KDM4ECYP3A4MAPTMEN1
SCHEMBL10893526 0.69 CA2 (0.55) CA2KDM4EMAPTMEN1KMT2A
SCHEMBL11043516 0.69 CA2 (0.62) CA2CYP3A4GAAMAPTKMT2A
SCHEMBL10545135 0.68 CA2 (0.61) CA2KDM4ECYP3A4MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4695634-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1987-09-22 US disclosed
US-4622406-A CHEMICAL INTERMEDIATES, TRIMETHYLSILOXY COMPOUNDS PFIZER INC. (US) 1986-11-11 US disclosed
US-4562267-A Intermediates of hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1985-12-31 US disclosed
US-4423233-A ALPHA-HYDROXY CARBOXIMIDATE INTERMEDIATES PFIZER INC. (US) 1983-12-27 US disclosed
US-4381308-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1983-04-26 US disclosed
US-4332952-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1982-06-01 US disclosed