SCHEMBL10763003

SCHEMBL10763003

Fc1ccc2nnc(S)n2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DYRK1A Q13627 2/20 0.33
DYRK2 Q92630 2/20 0.33
DYRK1B Q9Y463 1/20 0.32
HSD17B10 Q99714 3/20 0.31
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
PIM1 P11309 1/20 0.30
BRD4 O60885 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4247015 0.75 KDM4E (0.64) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL10026445 0.64 MET (0.47) KDM4EMEN1KMT2AHSD17B10BRD4
SCHEMBL2066171 0.64 DYRK1A (0.33) DYRK1ADYRK2DYRK1B
SCHEMBL11785295 0.64 MKNK1 (0.38) DYRK1A
SCHEMBL23642122 0.62 SCN5A (0.42) KDM4E
SCHEMBL9349085 0.57 RET (0.32) PIM1
SCHEMBL29394247 0.55
SCHEMBL2047395 0.55
SCHEMBL29142013 0.54 JAK2 (0.30) DYRK1ADYRK1B
SCHEMBL7158662 0.49

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0228061-A2 Cephem compounds Takeda Chemical Industries, Ltd. (JP) 1987-07-08 EP disclosed