Acacetin

Acacetin

SCHEMBL107712

COc1ccc(-c2cc(=O)c3c(O)cc(O)cc3o2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 6/20 1.00
MAPT P10636 6/20 1.00
CYP1A1 P04798 5/20 1.00
CYP1A2 P05177 5/20 1.00
MEN1 O00255 5/20 1.00
KMT2A Q03164 5/20 1.00
MAOB P27338 4/20 1.00
IP6K2 Q9UHH9 4/20 1.00
FLT3 P36888 4/20 1.00
NPC1 O15118 4/20 1.00
CYP3A4 P08684 4/20 1.00
CYP2C9 P11712 4/20 1.00
CYP2C19 P33261 4/20 1.00
ALDH1A1 P00352 4/20 1.00
MAOA P21397 4/20 1.00
TP53 P04637 3/20 1.00
CYP2D6 P10635 3/20 1.00
MAPK1 P28482 3/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
HIF1A Q16665 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acacetin SCHEMBL29387049 1.00 CYP1B1 (1.00) CYP1B1MAPTCYP1A1CYP1A2MEN1
Acacetin SCHEMBL28278297 0.99 CYP1B1 (0.97) CYP1B1MAPTCYP1A1CYP1A2MEN1
Apigenin Dimethylether SCHEMBL29392759 0.94 MAOB (1.00) CYP1B1MAPTCYP1A1CYP1A2MEN1
Apigenin Dimethylether SCHEMBL1176691 0.94 MAOB (1.00) CYP1B1MAPTCYP1A1CYP1A2MEN1
Acacetin SCHEMBL8304770 0.93 CYP1B1 (0.86) CYP1B1MAPTCYP1A1CYP1A2MEN1
Acacetin SCHEMBL8309340 0.93 CYP1B1 (0.86) CYP1B1MAPTCYP1A1CYP1A2MEN1
SCHEMBL30192733 0.89 CYP1B1 (0.80) CYP1B1MAPTCYP1A1CYP1A2MEN1
Genkwanin SCHEMBL29445006 0.89 FLT3 (1.00) CYP1B1MAPTCYP1A1CYP1A2MEN1
Apigenin SCHEMBL15475269 0.89 CYP1B1 (0.89) CYP1B1MAPTCYP1A1CYP1A2MEN1
Genkwanin SCHEMBL866123 0.89 FLT3 (1.00) CYP1B1MAPTCYP1A1CYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2745 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130395-A1 Water Dispersible Botanical Compositions AQUILA BLACK LTD (AU) 2026-05-14 US claimed
US-20260090969-A1 COMPOSITIONS THAT PROTECT CELLS FROM OXIDATIVE AND MITOCHONDRIAL STRESS Nuchido Limited (GB) 2026-04-02 US claimed
EP-4698662-A2 REGULATABLE CONTROLLED EXPRESSION OF A TRANSGENE IN PRIMATES AskBio Inc. (US) 2026-02-25 EP claimed
US-20250381166-A1 Cannabis-Derived Flavonoids And Related Methods CANURTA INC (CA) 2025-12-18 US claimed
US-20250367305-A1 ALBUMIN NANOCOMPOSITE COMPRISING PHYTOCHEMICAL AND COMPOSITION FOR IMPROVING MUSCLE DISEASE CONTAINING SAME SEOUL NATIONAL UNIVERSITY R&DB FOUNDATION (KR) 2025-12-04 US claimed
EP-4656062-A1 SALTY TASTE/UMAMI ENHANCER AJINOMOTO CO., INC. (JP) 2025-12-03 EP claimed
US-20250344731-A1 SALTY TASTE/UMAMI ENHANCER AJINOMOTO CO., INC. (JP) 2025-11-13 US claimed
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
US-20250212873-A1 VOLATILE HDAC INHIBITORS FOR THERAPEUTIC AND PLANT APPLICATIONS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-07-03 US claimed
WO-2024220449-A9 REGULATABLE CONTROLLED EXPRESSION OF A TRANSGENE IN PRIMATES AskBio Inc. (US) 2025-04-03 WO claimed
US-5958946-A APPLYING GLUCURONIC ACID GILLETTE COMPANY, THE (A DELAWARE CORPORATION) 1999-09-28 US claimed
WO-1999044578-A1 FORMULATIONS WITH AN ANTI-VIRAL EFFECT MERCK PATENT GMBH (DE) 1999-09-10 WO claimed
CN-1219102-A Process for propagation and/or selection of plant material SHELL INT RESEARCH (NL) 1999-06-09 CN claimed
US-5650433-A REDUCING ARTICULAR CARTILAGE DESTRUCTION IN A PATIENT BY ADMINISTERING A FLAVONOID COMPOUND KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1997-07-22 US claimed
EP-0633022-B1 Chondroprotective flavones KUREHA CHEMICAL IND CO LTD (JP) 1997-02-19 EP claimed
WO-1996031206-A2 FLAVONES AND COUMARINS AS AGENTS FOR THE TREATMENT OF ATHEROSCLEROSIS WARNER-LAMBERT COMPANY (US) 1996-10-10 WO claimed
CN-1100633-A Chondroprotective agents KUREHA CHEMICAL IND CO LTD (JP) 1995-03-29 CN claimed
EP-0633022-A2 Chondroprotective flavones KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-01-11 EP claimed
EP-0263553-A2 Method of inhibiting gene induction SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1988-04-13 EP claimed
US-4617293-A Flavonoid phosphate salts of aminoglycoside antibiotics MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1986-10-14 US claimed