SCHEMBL1077402

SCHEMBL1077402

COc1ccc(C2CNCc3cc(OCCCC4CCCNC4)ccc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.49
HRH3 Q9Y5N1 18/20 0.49
EED O75530 1/20 0.43
ACP1 P24666 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1037048 0.81 SLC6A4 (0.54) SLC6A4HRH3
SCHEMBL1034562 0.78 HRH3 (0.76) SLC6A4HRH3
SCHEMBL6715276 0.78 SLC6A4 (0.53) SLC6A4HRH3
SCHEMBL1035603 0.77 SLC6A4 (0.71) SLC6A4HRH3
SCHEMBL1077401 0.76 SLC6A4 (0.43) SLC6A4HRH3EED
Hydrochloric Acid SCHEMBL6632289 0.75 HRH3 (0.55) HRH3
SCHEMBL1035507 0.74 SLC6A4 (0.77) SLC6A4HRH3
SCHEMBL6614605 0.72 NPY1R (0.42) HRH3EEDACP1
SCHEMBL1036213 0.71 SLC6A4 (0.61) SLC6A4HRH3
SCHEMBL1034743 0.71 SLC6A4 (0.73) SLC6A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831173-B1 TETRAHYDROISOQUINOLINE COMPOUNDS FOR TREATMENT OF CNS DISORDERS JANSSEN PHARMACEUTICA NV (BE) 2011-01-26 EP disclosed