SCHEMBL10783166

SCHEMBL10783166

N#Cc1nc(Cl)c(Br)nc1N

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
GAA P10253 1/20 0.44
ALDH1A1 P00352 1/20 0.37
KHK P50053 1/20 0.35
USP8 P40818 1/20 0.34
CSNK1A1 P48729 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
MAPK14 Q16539 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10780291 0.92 ALDH1A1 (0.41) KDM4EGAAALDH1A1KHKUSP8
SCHEMBL10782113 0.82 USP8 (0.38) KDM4EUSP8SMN1; SMN2RXFP1
SCHEMBL10087543 0.82 ALDH1A1 (0.47) KDM4EGAAALDH1A1KHKUSP8
SCHEMBL29987465 0.82 ALDH1A1 (0.47) KDM4EGAAALDH1A1KHKUSP8
SCHEMBL3607648 0.80 KDM4E (0.44) KDM4EGAAALDH1A1KHKUSP8
SCHEMBL8200210 0.76 ALDH1A1 (0.45) KDM4EGAAALDH1A1KHKUSP8
SCHEMBL21074155 0.76 USP8 (0.37) USP8
SCHEMBL28965611 0.75 ALDH1A1 (0.41) KDM4EGAAALDH1A1KHKCSNK1A1
SCHEMBL11000333 0.75 KDM4E (0.40) KDM4EGAAALDH1A1KHKUSP8
SCHEMBL11117158 0.75 ALDH1A1 (0.46) KDM4EGAAALDH1A1KHKUSP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0132476-B1 ANTIMICROBIAL COMPOSITIONS MERCK & CO. INC. (US) 1987-07-15 EP disclosed
EP-0132476-A1 Antimicrobial compositions MERCK & CO. INC. (US) 1985-02-13 EP disclosed
US-4402959-A 3-AMINO-5,6-DIHALOPYRAZINE-2-CARBONITRILE MERCK & CO., INC. (US) 1983-09-06 US disclosed