SCHEMBL10784109

SCHEMBL10784109

CC(=O)NC(=O)Nc1ccc(S(=O)(=O)Oc2ccccc2)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
ALDH1A1 P00352 6/20 0.39
MAPT P10636 4/20 0.39
LMNA P02545 3/20 0.39
RECQL P46063 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 1/20 0.39
HSP90AA1 P07900 1/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
CA12 O43570 1/20 0.38
POLB P06746 2/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
ENPP3 O14638 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11521258 0.90 NPC1 (0.58) NPC1MEN1KMT2AALDH1A1MAPT
SCHEMBL11519736 0.88 NPC1 (0.43) NPC1MEN1KMT2AALDH1A1MAPT
SCHEMBL11521140 0.85 CA12 (0.52) NPC1MEN1KMT2AMAPTLMNA
SCHEMBL10784629 0.85 MEN1 (0.48) NPC1MEN1KMT2AMAPTLMNA
SCHEMBL11518679 0.85 DHODH (0.48) NPC1MEN1KMT2AALDH1A1MAPT
SCHEMBL11524372 0.84 NPC1 (0.42) NPC1MEN1KMT2AALDH1A1MAPT
SCHEMBL11519773 0.83 MEN1 (0.39) NPC1MEN1KMT2AMAPTLMNA
SCHEMBL10786890 0.83 ALDH1A1 (0.46) NPC1MEN1KMT2AALDH1A1MAPT
SCHEMBL11522204 0.81 POLB (0.47) MEN1KMT2AALDH1A1MAPTLMNA
SCHEMBL11519775 0.81 BDKRB1 (0.46) MEN1KMT2AMAPTKDM4ECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0105196-B1 SUBSTITUTED BENZENESULFONIC ACID ESTERS, PREPARATION THEREOF AND THEIR USE AS MEDICAMENTS HOECHST AKTIENGESELLSCHAFT (DE) 1987-07-29 EP disclosed
US-4504490-A Substituted benzenesulfonic esters and their use as medicaments for combatting helminths HOECHST AKTIENGESELLSCHAFT (DE) 1985-03-12 US disclosed
EP-0105196-A2 Substituted benzenesulfonic acid esters, preparation thereof and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1984-04-11 EP disclosed