SCHEMBL10784172

SCHEMBL10784172

O=C1NC2(CCOc3ccc(F)cc32)C(=O)N1CCCCCN1CCC(O)CC1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.46
MAPT P10636 2/20 0.46
AKR1B10 O60218 1/20 0.46
AKR1A1 P14550 1/20 0.46
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
SIGMAR1 Q99720 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10783302 0.99 AKR1B1 (0.47) AKR1B1MAPTAKR1B10AKR1A1ALDH1A1
SCHEMBL10783456 0.97 AKR1B1 (0.47) AKR1B1MAPTAKR1B10AKR1A1ALDH1A1
SCHEMBL10785899 0.87 KDM4E (0.44) MAPTALDH1A1GAA
SCHEMBL10787723 0.86 ALDH1A1 (0.41) MAPTALDH1A1GAASIGMAR1
SCHEMBL10787913 0.85 AKR1B1 (0.44) AKR1B1MAPTAKR1B10AKR1A1
SCHEMBL10785195 0.85 AKR1B1 (0.40) AKR1B1SIGMAR1
SCHEMBL10788567 0.85 SIGMAR1 (0.55) AKR1B1MAPTAKR1B10AKR1A1SIGMAR1
SCHEMBL10784811 0.84 KMT2A (0.41) ALDH1A1GAASIGMAR1
SCHEMBL10785027 0.84 AKR1B1 (0.40) AKR1B1SIGMAR1
SCHEMBL10520213 0.84 KMT2A (0.52) MAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4650798-A Antiarrhythmic 2,2-dialkyl-1-(aminoalkyl)-spiro[chroman-4,4'-imidazolidine]-2',5'-diones EISAI CO., LTD. (JP) 1987-03-17 US disclosed