SCHEMBL10784282

SCHEMBL10784282

CCn1c(=O)c2c(ncn2CCCCC(C)=O)n(C)c1=O

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 7/20 0.80
LMNA P02545 3/20 0.80
CYP1A2 P05177 2/20 0.80
NFKB1 P19838 2/20 0.80
ACHE P22303 2/20 0.80
PMP22 Q01453 2/20 0.80
ESR1 P03372 1/20 0.80
MAPT P10636 1/20 0.80
BLM P54132 1/20 0.80
RXFP1 Q9HBX9 2/20 0.77
MAPK1 P28482 1/20 0.77
ADORA2B P29275 7/20 0.68
PDE4B Q07343 6/20 0.68
PDE4C Q08493 6/20 0.68
PDE4D Q08499 6/20 0.68
TNF P01375 2/20 0.68
USP2 O75604 1/20 0.68
TSHR P16473 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
TRPA1 O75762 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802032 0.93 PDE4A (0.88) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL7800864 0.92 PDE4A (0.91) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL8362364 0.91 RXFP1 (0.67) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL11347084 0.91 PDE4A (0.89) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL11337820 0.91 PDE4A (0.89) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL10788889 0.91 PDE4A (0.89) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL11345748 0.91 PDE4A (0.89) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL10784646 0.90 PDE4A (0.84) PDE4ALMNACYP1A2NFKB1ACHE
SCHEMBL9682866 0.90 RXFP1 (0.77) PDE4ALMNACYP1A2NFKB1ACHE
Propentofylline SCHEMBL74602 0.89 PDE4A (1.00) PDE4ALMNACYP1A2NFKB1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0121439-B1 TRIS(DIALKYLAMINO)SULFONIUM BIFLUORIDE CATALYSTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1987-03-25 EP claimed
US-4636507-A Host defense mechanism enhancement HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-01-13 US claimed
EP-0121439-B1 TRIS(DIALKYLAMINO)SULFONIUM BIFLUORIDE CATALYSTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1987-03-25 EP disclosed
US-4598161-A Tris(dialkylamino)sulfonium bifluoride catalysts E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-07-01 US disclosed
EP-0121439-A1 Tris(dialkylamino)sulfonium bifluoride catalysts E.I. DU PONT DE NEMOURS AND COMPANY (US) 1984-10-10 EP disclosed