SCHEMBL9682866

SCHEMBL9682866

CC(=O)CCCCn1cnc2c1c(=O)n(CC(C)=O)c(=O)n2C

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.77
MAPK1 P28482 1/20 0.77
PDE4A P27815 5/20 0.77
LMNA P02545 3/20 0.77
CYP1A2 P05177 2/20 0.77
NFKB1 P19838 2/20 0.77
ACHE P22303 2/20 0.77
PMP22 Q01453 2/20 0.77
ESR1 P03372 1/20 0.77
MAPT P10636 1/20 0.77
BLM P54132 1/20 0.77
TRPA1 O75762 4/20 0.70
ADORA2B P29275 9/20 0.68
PDE4B Q07343 4/20 0.68
PDE4C Q08493 4/20 0.68
PDE4D Q08499 4/20 0.68
TNF P01375 2/20 0.68
USP2 O75604 1/20 0.68
TSHR P16473 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802032 0.93 PDE4A (0.88) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL9297147 0.90 PDE4A (0.80) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL10784282 0.90 PDE4A (0.80) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL7800864 0.89 PDE4A (0.91) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL11337820 0.88 PDE4A (0.89) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL10788889 0.88 PDE4A (0.89) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL11345748 0.88 PDE4A (0.89) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL11347084 0.88 PDE4A (0.89) RXFP1MAPK1PDE4ALMNACYP1A2
Lomifylline SCHEMBL1649451 0.87 RXFP1 (1.00) RXFP1MAPK1PDE4ALMNACYP1A2
SCHEMBL11401358 0.87 RXFP1 (0.72) RXFP1MAPK1PDE4ALMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082845-A Gastrointestinal HOECHST JAPAN LIMITED (JP) 1992-01-21 US disclosed
EP-0330031-B1 THERAPEUTIC AGENTS FOR THE TREATMENT OF PEPTIC ULCER DISEASE HOECHST JAPAN LIMITED (JP) 1991-12-11 EP disclosed
EP-0330031-A1 Therapeutic agents for the treatment of peptic ulcer disease HOECHST JAPAN LIMITED (JP) 1989-08-30 EP disclosed