SCHEMBL10791069

SCHEMBL10791069

CCOc1cc2c(C)nc(O)cc2cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
GAA P10253 2/20 0.56
ALDH1A1 P00352 1/20 0.56
RAC1 P63000 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
POLB P06746 1/20 0.48
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ENPP1 P22413 1/20 0.44
MAPT P10636 1/20 0.43
PDE3B Q13370 3/20 0.42
PDE3A Q14432 3/20 0.42
DPP4 P27487 2/20 0.41
PDE10A Q9Y233 1/20 0.39
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
CTSG P08311 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL149852 0.89 RAC1 (0.56) KDM4EGAAALDH1A1RAC1MEN1
SCHEMBL11971636 0.74 ALDH1A1 (0.57) KDM4EGAAALDH1A1RAC1MEN1
SCHEMBL11971491 0.72 HMGCR (0.45) KDM4EGAAALDH1A1RAC1MEN1
SCHEMBL9830708 0.72 MEN1 (0.44) KDM4EGAAALDH1A1MEN1KMT2A
SCHEMBL7846522 0.71 KDM4E (0.56) KDM4EGAAALDH1A1RAC1MEN1
SCHEMBL11971554 0.70 ALDH1A1 (0.42) KDM4EGAAALDH1A1RAC1MEN1
SCHEMBL28662301 0.70 KDM4E (0.57) KDM4EGAAENPP1MAPTPDE3B
SCHEMBL28311309 0.70 KDM4E (0.57) KDM4EGAAENPP1MAPTPDE3B
SCHEMBL15586088 0.70 ENPP1 (0.42) KDM4EGAAALDH1A1MEN1KMT2A
SCHEMBL24393297 0.69 ENPP1 (0.70) KDM4EALDH1A1ENPP1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4714705-A 4-nitrogen substituted isoquinolinol compounds having cardiotonic, phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1987-12-22 US disclosed