SCHEMBL1079779

SCHEMBL1079779

COc1ccccc1-n1c(-c2ccccc2)nc(C(N)=O)c1C

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
AVPR2 P30518 1/20 0.51
AVPR1A P37288 1/20 0.51
LMNA P02545 2/20 0.51
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 5/20 0.49
APOBEC3G Q9HC16 1/20 0.49
GLA P06280 2/20 0.48
THRB P10828 1/20 0.47
PTGS2 P35354 1/20 0.47
HPGD P15428 3/20 0.46
GAA P10253 2/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1076424 0.86 TSHR (0.51) TSHRAVPR2AVPR1ALMNAKDM4E
SCHEMBL1078087 0.82 NOTUM (0.47)
SCHEMBL16935851 0.77 AVPR2 (0.51) TSHRAVPR2AVPR1AKDM4EALDH1A1
SCHEMBL1076549 0.76 HTR2A (0.46) L3MBTL1
SCHEMBL28674639 0.70 ALDH1A1 (0.48) TSHRLMNAKDM4EALDH1A1THRB
SCHEMBL22289852 0.69 L3MBTL1 (0.53) TSHRAVPR2AVPR1AKDM4EALDH1A1
SCHEMBL28081745 0.69 AVPR2 (0.49) TSHRAVPR2AVPR1AKDM4EALDH1A1
SCHEMBL31532182 0.69 AVPR2 (0.55) TSHRAVPR2AVPR1AKDM4EALDH1A1
SCHEMBL21354520 0.68 GAA (0.56) TSHRAVPR2AVPR1ALMNAKDM4E
SCHEMBL16063426 0.68 CNR1 (0.54) TSHRLMNAKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005052-A2 NOVEL ARYLPIPERAZINE-CONTAINING IMIDAZOLE 4-CARBOXAMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME GREEN GROSS CORPORATION (KR) 2011-01-13 WO disclosed