SCHEMBL10798404

SCHEMBL10798404

CC(C)CN1C(N=Cc2ccc(Cl)cc2)=CC(=O)N2CCN=C21

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.38
ALDH1A1 P00352 3/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32
KMT2A Q03164 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
CNR1 P21554 1/20 0.31
CLPP Q16740 1/20 0.31
HTT P42858 1/20 0.31
NR1I2 O75469 1/20 0.30
HPGD P15428 1/20 0.30
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10798398 1.00 TSHR (0.38) TSHRALDH1A1MEN1CYP1A2MAPT
SCHEMBL11282584 0.84 TSHR (0.35) TSHRALDH1A1MEN1KMT2ATP53
SCHEMBL11282580 0.84 TSHR (0.35) TSHRALDH1A1MEN1KMT2ATP53
SCHEMBL10797980 0.74 TSHR (0.43) TSHRALDH1A1MAPTTP53CNR1
SCHEMBL10795887 0.72 LMNA (0.35) TSHRALDH1A1MEN1CYP1A2KMT2A
SCHEMBL10795455 0.67 TSHR (0.44) TSHRALDH1A1MAPTCYP2C9TP53
SCHEMBL10801005 0.64 TSHR (0.48) TSHRTP53GAACLPPHTT
SCHEMBL10800858 0.62 TSHR (0.33) TSHR
SCHEMBL10795740 0.59 TSHR (0.59) TSHRMEN1KMT2ATP53GAA
SCHEMBL11089172 0.57 ADORA2A (0.36) TSHRALDH1A1CYP1A2CLPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4642345-A BRONCHODILATOR AGENTS MEAD JOHNSON & COMPANY (US) 1987-02-10 US disclosed
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US disclosed
US-4404380-A BRONCHODILATORS, MEDIATOR RELEASE INHIBITORS, PHOSPHODIESTERASE INHIBITORS, AND VASODILATORS MEAD JOHNSON & COMPANY (US) 1983-09-13 US disclosed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US disclosed