SCHEMBL11089172

SCHEMBL11089172

CC(C)CN1C2=NCCN2C(=O)c2[nH]cnc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.36
ADORA2B P29275 2/20 0.36
TSHR P16473 5/20 0.34
PDE2A O00408 4/20 0.34
PDE1A P54750 4/20 0.34
PDE1B Q01064 4/20 0.34
PDE1C Q14123 4/20 0.34
CYP3A4 P08684 3/20 0.34
CFTR P13569 2/20 0.34
PDE5A O76074 1/20 0.34
CYP1A2 P05177 1/20 0.34
PDE4A P27815 1/20 0.34
MAPK1 P28482 1/20 0.34
ADORA1 P30542 1/20 0.34
SCN1A P35498 1/20 0.34
PDE6C P51160 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE3B Q13370 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018625 0.79 ALDH1A1 (0.32) TSHRPDE4AMAPK1PDE4BPDE4C
SCHEMBL6631440 0.78 LMNA (0.35) ADORA2AADORA2BTSHRPDE5APDE4A
SCHEMBL9585832 0.73 PDE4A (0.36) TSHRPDE4AMAPK1PDE4BPDE4C
SCHEMBL10800858 0.70 TSHR (0.33) TSHRCYP3A4SMN1; SMN2HIF1ALMNA
SCHEMBL10795887 0.68 LMNA (0.35) TSHRPDE2APDE1APDE1BPDE1C
SCHEMBL11063263 0.68 CYP3A4 (0.32) TSHRPDE2APDE1APDE1BPDE1C
SCHEMBL11273417 0.67 CYP3A4 (0.32) TSHRCYP3A4SMN1; SMN2HIF1A
SCHEMBL11074233 0.64 PDE4A (0.45) TSHRCYP1A2PDE4APDE4BPDE4C
SCHEMBL10801005 0.63 TSHR (0.48) TSHRCYP3A4PDE5APDE4AMAPK1
SCHEMBL10800120 0.63 MEN1 (0.49) ADORA2AADORA2BTSHRCYP1A2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US disclosed