SCHEMBL10798652

SCHEMBL10798652

CC1CN(CCN)CCC1Oc1nc2ccccc2n1Cc1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 10/20 0.49
CYP2D6 P10635 9/20 0.49
KCNH2 Q12809 8/20 0.49
CHRM1 P11229 4/20 0.49
EED O75530 2/20 0.49
SSTR5 P35346 4/20 0.47
TACR2 P21452 2/20 0.46
TACR1 P25103 2/20 0.46
MEN1 O00255 1/20 0.46
MLNR O43193 1/20 0.46
CACNA1F O60840 1/20 0.46
USP2 O75604 1/20 0.46
ABCB11 O95342 1/20 0.46
EGFR P00533 1/20 0.46
LMNA P02545 1/20 0.46
HLA-A P04439 1/20 0.46
ERBB2 P04626 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
LCK P06239 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10549456 1.00 HRH1 (0.49) HRH1CYP2D6KCNH2CHRM1EED
SCHEMBL9536666 1.00 HRH1 (0.49) HRH1CYP2D6KCNH2CHRM1EED
SCHEMBL9536973 0.86 EED (0.47) HRH1CYP2D6KCNH2CHRM1EED
SCHEMBL10549784 0.86 EED (0.47) HRH1CYP2D6KCNH2CHRM1EED
SCHEMBL10549770 0.86 EED (0.47) HRH1CYP2D6KCNH2CHRM1EED
SCHEMBL10548426 0.82 TP53 (0.49) HRH1CYP2D6KCNH2CHRM1SSTR5
SCHEMBL10799113 0.80 LMNA (0.51) HRH1CYP2D6KCNH2CHRM1EED
SCHEMBL9698401 0.80 SSTR5 (0.60) HRH1CYP2D6KCNH2CHRM1EED
Hydrochloric Acid SCHEMBL9537106 0.77 HRH1 (0.56) HRH1CYP2D6KCNH2CHRM1TP53
Hydrochloric Acid SCHEMBL9537102 0.77 HRH1 (0.56) HRH1CYP2D6KCNH2CHRM1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed