SCHEMBL10799321

SCHEMBL10799321

O=C1CCCC(=O)N1CCl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.42
POLB P06746 4/20 0.42
MEN1 O00255 3/20 0.42
PIK3CD O00329 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA1B P35368 1/20 0.33
GAA P10253 1/20 0.33
CA12 O43570 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112639 0.88
Hydrochloric Acid SCHEMBL28911779 0.77 POLB (0.47) KMT2APOLBMEN1CYP1A2CYP2C9
SCHEMBL6273408 0.75 MEN1 (0.55) KMT2APOLBMEN1CYP1A2CYP2C9
SCHEMBL14359370 0.74 POLB (0.53) KMT2APOLBMEN1BRD4BRD2
SCHEMBL719466 0.72 F2 (0.48) KMT2APOLBMEN1PIK3CDCHRM2
SCHEMBL6044381 0.72 KMT2A (0.42) KMT2APOLBMEN1PIK3CDCYP1A2
SCHEMBL8282999 0.72 KMT2A (0.42) KMT2APOLBMEN1PIK3CDCYP1A2
SCHEMBL9344572 0.72 KMT2A (0.42) KMT2APOLBMEN1PIK3CDCYP1A2
SCHEMBL7279979 0.72 KMT2A (0.42) KMT2APOLBMEN1PIK3CDCYP1A2
SCHEMBL717638 0.72 PIK3CD (0.57) KMT2APOLBMEN1PIK3CDBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4654433-A Process for the preparation of esters of amino acids MERCK & CO., INC. (US) 1987-03-31 US disclosed
US-4198413-A HYPOTENSIVE AGENTS MERCK & CO., INC. (US) 1980-04-15 US disclosed
US-4143146-A HYPOTENSIVE AGENTS MERCK & CO., INC. (US) 1979-03-06 US disclosed
US-4058530-A PHENYLALANINE, ANTIHYPERTENSIVE MERCK & CO., INC. (US) 1977-11-15 US disclosed
US-4051169-A HYPOTENSIVE AGENTS MERCK & CO., INC. (US) 1977-09-27 US disclosed
US-4038411-A ANTIHYPERTENSIVE AMINO ACID ESTERS MERCK & CO., INC. (US) 1977-07-26 US disclosed
US-3988341-A Esterification process MERCK & CO., INC. (US) 1976-10-26 US disclosed
US-3983138-A HYPOTENSIVES MERCK & CO., INC. (US) 1976-09-28 US disclosed