SCHEMBL10799731

SCHEMBL10799731

CCC(C(=O)c1ccc(Cl)cc1)n1cncn1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.48
CYP3A4 P08684 1/20 0.47
KMT2A Q03164 5/20 0.46
HSP90AA1 P07900 2/20 0.46
MEN1 O00255 3/20 0.45
MAPT P10636 2/20 0.43
LMNA P02545 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HTT P42858 3/20 0.42
POLB P06746 1/20 0.42
PDE4D Q08499 1/20 0.42
DNMT3A Q9Y6K1 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10469518 0.87 CYP3A4 (0.44) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL10418945 0.85 HSP90AA1 (0.48) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL10364784 0.84 KMT2A (0.54) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL6202493 0.82 MAPT (0.60) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL6227295 0.81 CYP19A1 (0.51) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL6203196 0.80 CYP3A4 (0.53) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL10468609 0.80 KMT2A (0.56) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL6222574 0.80 CYP19A1 (0.49) CYP19A1CYP3A4KMT2AMEN1MAPT
SCHEMBL9795408 0.80 CYP19A1 (0.53) CYP19A1CYP3A4KMT2AHSP90AA1MEN1
SCHEMBL11561868 0.79 KMT2A (0.49) CYP19A1CYP3A4KMT2AHSP90AA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0122693-B1 ANTIFUNGAL DI(AZOLYL)PROPANOL DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-08 EP disclosed
US-4625036-A Antifungal azole compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-11-25 US disclosed
EP-0122693-A1 Antifungal di(azolyl)propanol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-10-24 EP disclosed