SCHEMBL10799883

SCHEMBL10799883

Cc1ccc(S(=O)(=O)OCC2CCCCN2S(=O)(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 3/20 0.56
PSEN2 P49810 3/20 0.56
APH1B Q8WW43 3/20 0.56
NCSTN Q92542 3/20 0.56
APH1A Q96BI3 3/20 0.56
PSENEN Q9NZ42 3/20 0.56
TP53 P04637 1/20 0.54
TSHR P16473 1/20 0.54
CASP3 P42574 5/20 0.52
CASP7 P55210 4/20 0.52
CASP9 P55211 1/20 0.51
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
FKBP1A P62942 3/20 0.48
RAB9A P51151 1/20 0.48
PAX8 Q06710 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10799289 1.00 PSEN1 (0.56) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5337048 0.96 CASP3 (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8206528 0.96 CASP3 (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8206525 0.96 CASP3 (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12169307 0.85 CASP3 (0.64) CASP3CASP7CASP9RAB9APAX8
SCHEMBL15013036 0.85 CASP3 (0.64) CASP3CASP7CASP9RAB9APAX8
SCHEMBL15013035 0.85 CASP3 (0.64) CASP3CASP7CASP9RAB9APAX8
SCHEMBL10795608 0.83 PSEN1 (0.59) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9676145 0.83 HTR6 (0.46)
SCHEMBL10282723 0.83 PSEN1 (0.59) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4642348-A ANTIARRHYTHMIA AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1987-02-10 US disclosed
US-4593102-A N-[(amino)alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulfur linked substitution in the 2, 3 or 4-position A. H. ROBINS COMPANY, INC. (US) 1986-06-03 US disclosed
EP-0160436-A2 N-[(Amino)Alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulphur linked substitution in the 2, 3 or 4-position A.H. ROBINS COMPANY, INCORPORATED (US) 1985-11-06 EP disclosed