SCHEMBL10801656

SCHEMBL10801656

O=C(O)Cc1cc(F)ccc1Nc1c(Cl)cc(F)cc1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.61
CAMK2A Q9UQM7 3/20 0.60
ABCB11 O95342 2/20 0.55
PTGS1 P23219 2/20 0.55
NR1I3 Q14994 2/20 0.55
PPARG P37231 1/20 0.55
CXCL8 P10145 3/20 0.54
TTR P02766 2/20 0.54
AKR1B10 O60218 1/20 0.54
UGT1A9 O60656 1/20 0.54
TRPA1 O75762 1/20 0.54
MT-CO2 P00403 1/20 0.54
ALB P02768 1/20 0.54
UGT1A6 P19224 1/20 0.54
UGT1A1 P22309 1/20 0.54
CXCR1 P25024 1/20 0.54
ADRA1A P35348 1/20 0.54
AGTR2 P50052 1/20 0.54
SLC22A6 Q4U2R8 1/20 0.54
NR1H4 Q96RI1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10796562 0.90 CAMK2A (0.75) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL10797038 0.86 CAMK2A (0.77) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL1033041 0.82 PTGS2 (0.71) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL1031441 0.82 PTGS2 (0.74) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL1032030 0.80 PTGS2 (0.56) PTGS2CAMK2AABCB11PTGS1NR1I3
4',5-Dihydroxy-Diclofenac SCHEMBL7162002 0.79 CAMK2A (0.81) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL1032830 0.79 PTGS2 (0.54) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL1032535 0.77 PTGS2 (0.87) PTGS2CAMK2AABCB11PTGS1NR1I3
Lumiracoxib SCHEMBL6063194 0.76 PTGS2 (0.87) PTGS2CAMK2AABCB11PTGS1NR1I3
SCHEMBL30911087 0.76 MEN1 (0.52) CAMK2ACXCL8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4711879-A IMMUNO-MODULATING ACTIVITY CIBA-GEIGY CORPORATION (US) 1987-12-08 US claimed
US-4640911-A IMMUNOSTIMULANTS, VIRICIDES SUCH AS HERPES SIMPLEX CIBA-GEIGY CORPORATION (US) 1987-02-03 US claimed
EP-0163286-A2 Acylated sugars, method for their preparation and their use CIBA-GEIGY AG (CH) 1985-12-04 EP claimed
US-4640911-A IMMUNOSTIMULANTS, VIRICIDES SUCH AS HERPES SIMPLEX CIBA-GEIGY CORPORATION (US) 1987-02-03 US disclosed