SCHEMBL10808985

SCHEMBL10808985

CCCC(=O)C1=NC(=O)N=C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.37
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
FASN P49327 1/20 0.32
LMNA P02545 2/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
STS P08842 1/20 0.30
FFAR3 O14843 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26254861 0.60 HSD17B3 (0.82) HSD17B3HPGDALDH1A1RECQLTDP1
SCHEMBL26254903 0.60 HSD17B3 (0.48) HSD17B3HPGDALDH1A1ALOX15TSHR
Propyl 4-Pyridyl Ketone SCHEMBL4952700 0.57 HSD17B3 (0.61) HSD17B3HPGDALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL3346960 0.56 CTNNB1 (0.58) HPGDALDH1A1ALOX15TSHRRECQL
SCHEMBL7195006 0.56 HSD17B3 (0.64) HSD17B3HPGDALDH1A1SMN1; SMN2L3MBTL1
Butyrophenone SCHEMBL25423577 0.56 L3MBTL1 (0.77) HSD17B3HPGDALDH1A1ALOX15TDP1
SCHEMBL19457972 0.56 HSD17B3 (0.48) HSD17B3HPGDALDH1A1ALOX15TSHR
Butyrophenone SCHEMBL82532 0.56 L3MBTL1 (0.77) HSD17B3HPGDALDH1A1ALOX15TDP1
Butyrophenone SCHEMBL9725428 0.56 L3MBTL1 (0.77) HSD17B3HPGDALDH1A1ALOX15TDP1
Butyrophenone SCHEMBL11522791 0.56 L3MBTL1 (0.77) HSD17B3HPGDALDH1A1ALOX15TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0079049-B1 NOVEL SUBSTITUTED ALKANOYLIMIDAZOL-2-ONE DERIVATIVES MERRELL DOW PHARMACEUTICALS INC. (US) 1987-04-01 EP disclosed
US-4447619-A CARDIOTONIC AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1984-05-08 US disclosed
EP-0079049-A2 Novel substituted alkanoylimidazol-2-one derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1983-05-18 EP disclosed
US-4367236-A CARDIOTONIC AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1983-01-04 US disclosed