SCHEMBL10810325

SCHEMBL10810325

COc1ccc2nc(NC(N)=S)sc2c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 12/20 0.72
RAB9A P51151 12/20 0.72
MEN1 O00255 7/20 0.72
KMT2A Q03164 7/20 0.72
MAPT P10636 7/20 0.72
ALDH1A1 P00352 5/20 0.72
HTT P42858 3/20 0.72
NFKB1 P19838 3/20 0.72
NFKB2 Q00653 3/20 0.72
RELA Q04206 3/20 0.72
LMNA P02545 2/20 0.72
HPGD P15428 1/20 0.72
MPI P34949 1/20 0.72
NPSR1 Q6W5P4 1/20 0.72
APOBEC3G Q9HC16 1/20 0.72
TDP1 Q9NUW8 1/20 0.72
SMN1; SMN2 Q16637 8/20 0.69
CYP1A2 P05177 1/20 0.69
CYP3A4 P08684 1/20 0.69
CYP2C19 P33261 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10804473 0.86 NPC1 (0.69) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL23715 0.82 NPC1 (0.70) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL4918595 0.82 NPC1 (1.00) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL15993384 0.81 DYRK1A (0.67) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2114859 0.81 NPC1 (0.68) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL10807219 0.81 NPC1 (0.74) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL1307056 0.81 MAPT (0.82) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL5653636 0.80 CASP2 (0.77) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL16681363 0.80 SCD (0.88) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL11549742 0.80 NPC1 (0.76) NPC1RAB9AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0093515-B1 TRICYCLIC TRIAZINO COMPOUNDS, THEIR USE AND FORMULATION AS PHARMACEUTICALS AND PROCESSES FOR THEIR PRODUCTION FISONS plc (GB) 1987-01-21 EP disclosed
US-4499269-A IMMUNO-REGULANT, SKIN DISORDERS, ANTITUMOR AGENTS FISONS PLC (GB) 1985-02-12 US disclosed
EP-0093515-A1 Tricyclic triazino compounds, their use and formulation as pharmaceuticals and processes for their production FISONS plc (GB) 1983-11-09 EP disclosed