SCHEMBL1081985

SCHEMBL1081985

COC(=O)CC1c2[nH]c3ccc(-c4noc(-c5cc(Cl)nc(OC)c5)n4)cc3c2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 9/20 0.44
S1PR4 O95977 1/20 0.40
S1PR5 Q9H228 1/20 0.40
BRD3 Q15059 2/20 0.34
ABCG2 Q9UNQ0 2/20 0.33
TP53 P04637 3/20 0.33
MAPT P10636 3/20 0.33
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
ABCB1 P08183 1/20 0.32
TBK1 Q9UHD2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL948464 0.91 S1PR1 (0.48) S1PR1S1PR4S1PR5ABCG2TP53
SCHEMBL946662 0.87 S1PR1 (0.58) S1PR1S1PR4S1PR5
Hydrochloric Acid SCHEMBL946955 0.80 S1PR1 (0.49) S1PR1S1PR4S1PR5
SCHEMBL2567415 0.77 S1PR1 (0.70) S1PR1S1PR4S1PR5
SCHEMBL2563713 0.76 S1PR1 (0.58) S1PR1S1PR4S1PR5MAPTTLR8
SCHEMBL944763 0.76 TRPV1 (0.50) BRD3TP53MAPTSIRT1
SCHEMBL946049 0.76 S1PR1 (0.56) S1PR1S1PR4S1PR5
SCHEMBL947736 0.73 SLC6A4 (0.42) BRD3ABCG2TP53MAPTSMN1; SMN2
SCHEMBL948216 0.73 S1PR1 (0.69) S1PR1S1PR4S1PR5
SCHEMBL949317 0.73 BRD3 (0.40) BRD3ABCG2TP53MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed