SCHEMBL10823218

SCHEMBL10823218

CC(C)(CC(=O)CO[PH](=O)O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.42
HIF1A Q16665 1/20 0.42
TAAR1 Q96RJ0 1/20 0.38
ME2 P23368 2/20 0.37
ME1 P48163 2/20 0.37
ME3 Q16798 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNN4 O15554 1/20 0.35
ALOX15 P16050 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10823220 0.90 CYP2C19 (0.44) CYP2C19HIF1ATAAR1ME2ME1
SCHEMBL10823234 0.80 GAA (0.31) NPC1RAB9AGAA
SCHEMBL7207085 0.78 CYP2C19 (0.42) CYP2C19HIF1ATAAR1ME2ME1
SCHEMBL10823000 0.78 KMT2A (0.46) CYP2C19HIF1AALDH1A1MAPTKMT2A
SCHEMBL6918240 0.77 GPR55 (0.37) HIF1AALDH1A1HTTMAPTKMT2A
SCHEMBL873147 0.74 CYP2C19 (0.52) CYP2C19HIF1ATAAR1ME2ME1
SCHEMBL29113204 0.74
SCHEMBL32663593 0.73 CYP2C19 (0.40) CYP2C19HIF1AALDH1A1MAPTKMT2A
SCHEMBL57411 0.72 CYP2C19 (0.69) CYP2C19HIF1ATAAR1ME2ME1
SCHEMBL16964970 0.71 CES1 (0.47) HIF1AALDH1A1KMT2AHDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0089769-B1 9-SUBSTITUTED CARBACYCLIN ANALOGUES THE UPJOHN COMPANY (US) 1986-10-01 EP disclosed
US-4611005-A BRONCHODILATORS, ASTHMA, ANTICOAGULANTS E. R. SQUIBB & SONS, INC. (US) 1986-09-09 US disclosed
EP-0092352-B1 9-SUBSTITUTED CARBACYCLINS THE UPJOHN COMPANY (US) 1986-07-02 EP disclosed
EP-0086611-B1 9-SUBSTITUTED CARBACYCLIN ANALOGUES THE UPJOHN COMPANY (US) 1986-05-21 EP disclosed
US-4588823-A 9-substituted carbacyclin analogs THE UPJOHN COMPANY (US) 1986-05-13 US disclosed
US-4585886-A 9-Substituted carbacyclin analogs THE UPJOHN COMPANY (US) 1986-04-29 US disclosed
US-4490555-A 9-Substituted carbacyclin analogs THE UPJOHN COMPANY (US) 1984-12-25 US disclosed
US-4487960-A 9-Substituted carbacyclin analogs THE UPJOHN COMPANY (US) 1984-12-11 US disclosed
US-4487961-A ANTIULCER, ANTIASTHMA, ANTICOAGULANTS THE UPJOHN COMPANY (US) 1984-12-11 US disclosed
EP-0092352-A1 9-Substituted carbacyclins THE UPJOHN COMPANY (US) 1983-10-26 EP disclosed
EP-0089769-A1 9-Substituted carbacyclin analogues THE UPJOHN COMPANY (US) 1983-09-28 EP disclosed
EP-0086611-A1 9-Substituted carbacyclin analogues THE UPJOHN COMPANY (US) 1983-08-24 EP disclosed
US-4028350-A ANTIINFLAMMATORY AGENTS THE UPJOHN COMPANY (US) 1977-06-07 US disclosed