SCHEMBL10825083

SCHEMBL10825083

COC(=O)[C@@H](C)N[C@@H](CC(C)(C)C)C(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.51
CTSL P07711 1/20 0.51
CTSB P07858 1/20 0.51
MAPT P10636 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 3/20 0.43
CAPN1 P07384 1/20 0.43
POLB P06746 1/20 0.42
ALOX15 P16050 1/20 0.42
KYNU Q16719 1/20 0.41
CTSK P43235 3/20 0.41
TACR1 P25103 1/20 0.41
THRB P10828 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10705812 1.00 CTSS (0.51) CTSSCTSLCTSBMAPTL3MBTL1
SCHEMBL10706806 0.84 CAPN1 (0.55) CTSSCTSLCTSBCAPN1CTSK
SCHEMBL10825080 0.84 CAPN1 (0.55) CTSSCTSLCTSBCAPN1CTSK
SCHEMBL10706801 0.84 CAPN1 (0.55) CTSSCTSLCTSBCAPN1CTSK
SCHEMBL3044553 0.78 CTSS (0.70) CTSSCTSLCTSBALDH1A1ALOX15
SCHEMBL13295150 0.78 CTSS (0.56) CTSSCTSLCTSBALDH1A1ALOX15
SCHEMBL22692566 0.78 ALDH1A1 (0.58) CTSSCTSLCTSBMAPTL3MBTL1
SCHEMBL21078552 0.78 MAPT (0.50) CTSSCTSLCTSBMAPTL3MBTL1
SCHEMBL23008679 0.77 ALDH1A1 (0.53) CTSSCTSLCTSBL3MBTL1ALDH1A1
SCHEMBL4395801 0.76 ACE (0.51) L3MBTL1ALOX15CTSKHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4568666-A COLLAGENASE INHIBITORS, ANTIARTJRITIC AGENTS G. D. SEARLE & CO. (US) 1986-02-04 US disclosed
US-4511504-A COLLAGENASE INHIBITORS G.D. SEARLE & CO. (US) 1985-04-16 US disclosed
EP-0126974-A1 Carboxyalkyl peptide derivatives G.D. Searle & Co. (US) 1984-12-05 EP disclosed