SCHEMBL10825239

SCHEMBL10825239

CC(C)(C)OC(=O)C[C@H](NC1CCCCC1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 3/20 0.43
GAA P10253 1/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC4 P56524 1/20 0.40
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
BTK Q06187 1/20 0.38
EPHX2 P34913 1/20 0.38
CACNA1B Q00975 4/20 0.36
LMNA P02545 1/20 0.36
CYP2D6 P10635 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19744864 1.00 EPHX1 (0.43) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL38057 0.98 EPHX1 (0.40) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL38058 0.98 EPHX1 (0.40) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL38034 0.85 EPHX1 (0.40) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL38032 0.85 EPHX1 (0.40) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL29401399 0.82 HDAC4 (0.49) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL3311032 0.82 HDAC4 (0.49) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL27996141 0.82 HDAC4 (0.49) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL24033741 0.82 EPHX1 (0.44) EPHX1GAAHDAC1HDAC6HDAC4
SCHEMBL24033578 0.82 EPHX1 (0.44) EPHX1GAAHDAC1HDAC6HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4603121-A ANALGESICS G. D. SEARLE & CO. (US) 1986-07-29 US disclosed
US-4514332-A Tetrapeptide adamantyl amides G. D. SEARLE & CO. (US) 1985-04-30 US disclosed
EP-0136720-A2 Enkephalin analogs G.D. Searle & Co. (US) 1985-04-10 EP disclosed
US-4495178-A Enkephalin analogs G. D. SEARLE & CO. (US) 1985-01-22 US disclosed