SCHEMBL10828486

SCHEMBL10828486

COC(=O)Cc1nc(NC=O)cc(OC)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
CYP1A2 P05177 2/20 0.36
KMT2A Q03164 2/20 0.36
ADORA3 P0DMS8 2/20 0.36
ADORA1 P30542 1/20 0.35
HSP90AB1 P08238 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8686002 0.83 CYP1A2 (0.50) ALDH1A1KDM4ECYP1A2KMT2AHSP90AB1
SCHEMBL15317599 0.77 ALDH1A1 (0.43) ALDH1A1KDM4ECYP1A2KMT2AHSP90AB1
SCHEMBL9461045 0.77 ALDH1A1 (0.48) ALDH1A1KDM4ECYP1A2HSP90AB1SMN1; SMN2
SCHEMBL10828626 0.76 ALDH1A1 (0.42) ALDH1A1KDM4ECYP1A2HSP90AB1SMN1; SMN2
SCHEMBL10828739 0.74 KDM4E (0.39) ALDH1A1KDM4ECYP1A2KMT2AHSP90AB1
SCHEMBL10828437 0.74 KDM4E (0.40) ALDH1A1KDM4ECYP1A2KMT2ASMN1; SMN2
SCHEMBL8687010 0.72 KDM4E (0.49) ALDH1A1KDM4ECYP1A2KMT2ASMN1; SMN2
SCHEMBL5092329 0.69 CYP1A2 (0.48) ALDH1A1KDM4EL3MBTL1CYP1A2KMT2A
SCHEMBL24759680 0.68 MTNR1A (0.46) ALDH1A1KDM4EHSP90AB1SMN1; SMN2
SCHEMBL8687107 0.68 TSHR (0.45) ALDH1A1KDM4EL3MBTL1CYP1A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4596869-A Pyridinyl and pyrimidinyl derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1986-06-24 US disclosed
US-4395411-A ANTIBIOTICS; BACTERICIDES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-07-26 US disclosed
US-4267176-A Amino or acylamino-substituted pyrimidinyl cephalosporanic acid derivatives and pharmaceutical compositions thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-05-12 US disclosed