SCHEMBL10832004

SCHEMBL10832004

CN(C)CCNc1ccccc1C#N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.53
TSHR P16473 3/20 0.53
HPGD P15428 3/20 0.53
HSD17B10 Q99714 2/20 0.53
CYP2C19 P33261 1/20 0.44
NCF1 P14598 2/20 0.43
GAA P10253 3/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
SLC2A1 P11166 1/20 0.41
ALDH1A1 P00352 4/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
MALT1 Q9UDY8 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14662152 0.83 CYP2C19 (0.44) KDM4ECYP2C19NCF1GAASLC2A1
SCHEMBL14670113 0.83 CYP2C19 (0.44) KDM4ECYP2C19NCF1GAASLC2A1
SCHEMBL2122821 0.80 TSHR (0.58) KDM4ETSHRHPGDHSD17B10GAA
SCHEMBL28317278 0.79 NCF1 (0.40) KDM4EHPGDNCF1GAASLC2A1
SCHEMBL9025129 0.78 NCF1 (0.42) KDM4EHPGDNCF1SLC2A1ALDH1A1
SCHEMBL10831149 0.78 TSHR (0.47) KDM4ETSHRHPGDHSD17B10GAA
SCHEMBL10831309 0.78 KDM4E (0.47) KDM4ETSHRHPGDHSD17B10GAA
SCHEMBL30528606 0.77 TSHR (0.56) KDM4ETSHRHPGDHSD17B10CYP2C19
SCHEMBL3568604 0.77 TSHR (0.56) KDM4ETSHRHPGDHSD17B10CYP2C19
SCHEMBL20156858 0.77 TSHR (0.58) KDM4ETSHRHPGDHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4585869-A ANTIINFLAMMATORY, ANALGESIC, ANTIULCER ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1986-04-29 US disclosed
US-4549023-A ANTINFLAMMATORY AGENTS, ANALGESICS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1985-10-22 US disclosed
US-4474964-A 3-Aminoindazole derivatives ASAHI, KASEI, KOGYO, KABUSHIKI, KAISHA (JP) 1984-10-02 US disclosed
EP-0049779-A1 3-Aminoindazole derivatives and process for preparation thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-04-21 EP disclosed