SCHEMBL10835784

SCHEMBL10835784

Oc1cnn(-c2ccc(Cl)cc2F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
EPHX2 P34913 1/20 0.40
RAB9A P51151 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
GRM5 P41594 1/20 0.34
NOTUM Q6P988 1/20 0.34
TRPM5 Q9NZQ8 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNH2 Q12809 1/20 0.34
CCR2 P41597 2/20 0.33
SCN9A Q15858 1/20 0.33
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10835575 0.83 NOTUM (0.49) GAAEPHX2NOTUMCYP3A4KCNH2
SCHEMBL7222099 0.81 GAA (0.42) GAAEPHX2GRM5NOTUMJAK2
SCHEMBL12989360 0.81 ESR1 (0.40) GAAMEN1KMT2AKCNH2
SCHEMBL23302371 0.78 EPHX2 (0.58) GAAEPHX2RAB9AMEN1KMT2A
SCHEMBL28890862 0.78 TRPM5 (0.35) GRM5NOTUMTRPM5CYP1A2CYP3A4
SCHEMBL2417589 0.72 GAA (0.66) GAAEPHX2RAB9ANOTUMMEN1
SCHEMBL12988811 0.71 TDO2 (0.41) RAB9AMEN1KMT2ACYP1A2CYP3A4
SCHEMBL25113382 0.71 CYP3A4 (0.46) RAB9AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL10950640 0.70 GAA (0.63) GAAEPHX2RAB9ANOTUMMEN1
SCHEMBL30719692 0.70 NOTUM (0.53) GAANOTUMMEN1KMT2AJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4621144-A 1-phenyl-4-hydroxypyrazole derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-11-04 US claimed