SCHEMBL10844142

SCHEMBL10844142

c1cn(CCC2CCCNCC2)cn1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.49
TBXAS1 P24557 8/20 0.42
CYP19A1 P11511 5/20 0.42
HRH3 Q9Y5N1 2/20 0.40
HRH4 Q9H3N8 1/20 0.40
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
FDPS P14324 1/20 0.38
GAA P10253 1/20 0.36
QPCT Q16769 1/20 0.36
EGLN3 Q9H6Z9 1/20 0.36
PIM1 P11309 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8164980 0.94 CYP2B6 (0.46) CYP2B6TBXAS1CYP19A1HRH3HRH4
Hydrochloric Acid SCHEMBL10845833 0.91 CYP2B6 (0.44) CYP2B6TBXAS1CYP19A1HRH3CYP11B1
SCHEMBL6174188 0.84 TBXAS1 (0.52) CYP2B6TBXAS1CYP19A1HRH3HRH4
SCHEMBL11051486 0.84 CYP2B6 (0.68) CYP2B6TBXAS1CYP19A1HRH3HRH4
SCHEMBL11050188 0.84 CYP2B6 (0.68) CYP2B6TBXAS1CYP19A1HRH3HRH4
Iodide SCHEMBL16164357 0.82 CYP2B6 (0.66) CYP2B6TBXAS1CYP19A1HRH3HRH4
SCHEMBL13350294 0.82 TBXAS1 (0.54) CYP2B6TBXAS1CYP19A1HRH3HRH4
SCHEMBL1088292 0.77 CYP2B6 (0.68) CYP2B6TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL18505978 0.77 TBXAS1 (0.48) CYP2B6TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL11047220 0.76 CYP2B6 (0.61) CYP2B6TBXAS1CYP19A1HRH3HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4605744-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1986-08-12 US disclosed
US-4537969-A AZOLE-SUBSTITUTED SATURATED HETEROCYCLIC CARBOXALDEHYDE ACETALS;INTERMEDIATES FOR 6-AMIDINOPENICILLINS HOFFMANN-LA ROCHE INC. (US) 1985-08-27 US disclosed
EP-0148283-A1 Novel penicillanic acid derivatives F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-07-17 EP disclosed
US-4431653-A ANTIBIOTICS; BACTERICIDES; SSYNERGISTIC WITH AMINO ACID DERIVATIVE HOFFMANN-LA ROCHE INC. (US) 1984-02-14 US disclosed