SCHEMBL11047220

SCHEMBL11047220

c1cn(CCCC2CCCC2)cn1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.61
TBXAS1 P24557 10/20 0.57
HRH4 Q9H3N8 1/20 0.53
HRH3 Q9Y5N1 1/20 0.53
CYP19A1 P11511 5/20 0.49
GAA P10253 1/20 0.49
QPCT Q16769 1/20 0.49
PRKCI P41743 1/20 0.44
TPSAB1 Q15661 1/20 0.43
TPSD1 Q9BZJ3 1/20 0.43
TPSG1 Q9NRR2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24833975 0.98 CYP2B6 (0.64) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL11049587 0.98 CYP2B6 (0.64) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL16163635 0.93 CYP2B6 (0.62) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL11051486 0.87 CYP2B6 (0.68) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL11050188 0.87 CYP2B6 (0.68) CYP2B6TBXAS1HRH4HRH3CYP19A1
Iodide SCHEMBL16164357 0.86 CYP2B6 (0.66) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL24833961 0.85 CYP2B6 (0.53) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL10784468 0.85 TBXAS1 (0.49) CYP2B6TBXAS1HRH4HRH3GAA
SCHEMBL6174188 0.85 TBXAS1 (0.52) CYP2B6TBXAS1HRH4HRH3CYP19A1
SCHEMBL11720830 0.82 TBXAS1 (0.53) CYP2B6TBXAS1HRH4HRH3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000951-B1 PHARMACEUTICAL FORMULATIONS COMPRISING 1-SUBSTITUTED IMIDAZOLES, 1-SUBSTITUTED IMIDAZOLES AND 1-SUBSTITUTED IMIDAZOLES FOR USE IN THE TREATMENT OR PROPHYLAXIS OF THROMBO-EMBOLIC DISORDERS THE WELLCOME FOUNDATION LIMITED (GB) 1984-05-23 EP disclosed
EP-0000950-B1 IMIDAZOLE DERIVATIVES AND SALTS THEREOF AND THEIR SYNTHESIS THE WELLCOME FOUNDATION LIMITED (GB) 1984-02-01 EP disclosed
US-4317830-A ANTISHOCK AGENTS, ANTICOAGULANTS BURROUGHS WELLCOME CO. (US) 1982-03-02 US disclosed
US-4284641-A ANTITHROMBOEMBOLIC AGENT BURROUGHS WELLCOME CO. (US) 1981-08-18 US disclosed
EP-0000950-A1 Imidazole derivatives and salts thereof and their synthesis THE WELLCOME FOUNDATION LIMITED (GB) 1979-03-07 EP disclosed
EP-0000951-A1 Pharmaceutical Formulations comprising 1-substituted imidazoles, 1-substituted imidazoles and 1-substituted imidazoles for use in the treatment or prophylaxis of thrombo-embolic disorders THE WELLCOME FOUNDATION LIMITED (GB) 1979-03-07 EP disclosed