SCHEMBL10864396

SCHEMBL10864396

COc1ccccc1N1CCN(CCCCCc2ccc(OC)c(S(N)(=O)=O)c2)CC1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.60
HTR2C P28335 4/20 0.60
DRD2 P14416 3/20 0.56
DRD3 P35462 1/20 0.54
MEN1 O00255 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HTR7 P34969 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10865028 0.99 HTR1A (0.59) HTR1AHTR2CDRD2DRD3MEN1
SCHEMBL10863541 0.92 HTR1A (0.52) HTR1AHTR2CDRD2DRD3HTR7
SCHEMBL10864701 0.91 HTR1A (0.58) HTR1AHTR2CDRD2DRD3MEN1
Hydrochloric Acid SCHEMBL10864557 0.91 HTR1A (0.51) HTR1AHTR2CDRD2DRD3
SCHEMBL10864089 0.90 HTR1A (0.56) HTR1AHTR2CDRD2DRD3
SCHEMBL10863803 0.89 SIGMAR1 (0.53) HTR2CDRD2DRD3HTR7
SCHEMBL10863723 0.88 HTR1A (0.54) HTR1AHTR2CDRD2DRD3HTR7
SCHEMBL10966019 0.82 HTR1A (0.58) HTR1AHTR2CDRD2DRD3HTR7
SCHEMBL10864387 0.82 DRD4 (0.68) HTR1ADRD2KMT2A
Hydrochloric Acid SCHEMBL10865378 0.82 HTR1A (0.58) HTR1AHTR2CDRD2DRD3HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4613598-A HYPOTENSIVE AGENTS MITSUBISHI CHEMICAL INDUSTRIES LIMITED (JP) 1986-09-23 US disclosed
EP-0154969-A2 Piperazine derivatives and their acid addition salts MITSUBISHI KASEI CORPORATION (JP) 1985-09-18 EP disclosed