SCHEMBL10864591

SCHEMBL10864591

Clc1ccc2nc(-c3ccccc3)cc(Cl)c2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.65
AURKA O14965 1/20 0.58
AURKB Q96GD4 1/20 0.58
ESRRB O95718 1/20 0.58
ESR1 P03372 1/20 0.58
ESRRA P11474 1/20 0.58
ESR2 Q92731 1/20 0.58
ALDH1A1 P00352 3/20 0.54
HPGD P15428 3/20 0.54
PTGES O14684 1/20 0.54
ALOX5 P09917 1/20 0.54
CYP2C9 P11712 1/20 0.54
CASP7 P55210 1/20 0.54
HIF1A Q16665 1/20 0.54
HSD17B10 Q99714 1/20 0.54
ELANE P08246 1/20 0.54
ADORA1 P30542 1/20 0.51
DHODH Q02127 3/20 0.51
MAPT P10636 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10865179 0.91 ESR1 (0.65) MAPK1AURKAAURKBESRRBESR1
SCHEMBL6534510 0.88 MAPK1 (0.55) MAPK1AURKAAURKBESRRBESR1
SCHEMBL8956330 0.86 MAPK1 (0.85) MAPK1AURKAAURKBALDH1A1HPGD
SCHEMBL10865067 0.85 DHODH (0.68) MAPK1AURKAAURKBESRRBESR1
SCHEMBL10864870 0.85 DHODH (0.68) MAPK1AURKAAURKBESRRBESR1
SCHEMBL8410911 0.84 MAPK1 (0.82) MAPK1AURKAAURKBESR1ESR2
SCHEMBL785473 0.83 ACHE (0.61) MAPK1ESRRBESR1ESRRAESR2
SCHEMBL29793367 0.83 ACHE (0.61) MAPK1ESRRBESR1ESRRAESR2
SCHEMBL10864863 0.83 DHODH (0.58) MAPK1ESRRBESR1ESRRAESR2
SCHEMBL10865512 0.83 LMNA (0.62) MAPK1ESRRBESR1ESRRAESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0168812-A1 4-Amino-2-phenyl quinolines, methods and intermediates for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1986-01-22 EP disclosed
US-4560692-A ANTICONVULSANTS OR ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1985-12-24 US disclosed