SCHEMBL10865646

SCHEMBL10865646

CN(C)S(=O)(=O)c1cc(C(=O)CCCCN2CCN(c3ccccc3)CC2)ccc1S(C)(=O)=O

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.48
HTR7 P34969 3/20 0.48
DRD4 P21917 4/20 0.47
DRD2 P14416 3/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
SLC6A4 P31645 1/20 0.47
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10865051 0.99 DRD4 (0.48) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10863098 0.97 THRA (0.47) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10863523 0.88 HTR1A (0.50) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10864609 0.87 DRD4 (0.49) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10864507 0.87 HTR1A (0.45) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10864514 0.87 DRD4 (0.52) HTR1ADRD4DRD2GAA
SCHEMBL10865808 0.87 HTR1A (0.48) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10863236 0.86 HTR1A (0.48) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10864154 0.86 DRD4 (0.45) HTR1AHTR7DRD4DRD2HTR2A
SCHEMBL10865638 0.86 DRD4 (0.53) HTR1ADRD4DRD2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4613598-A HYPOTENSIVE AGENTS MITSUBISHI CHEMICAL INDUSTRIES LIMITED (JP) 1986-09-23 US disclosed
EP-0154969-A2 Piperazine derivatives and their acid addition salts MITSUBISHI KASEI CORPORATION (JP) 1985-09-18 EP disclosed