SCHEMBL10882913

SCHEMBL10882913

COc1ccc(C(=O)Nc2ccc(OCC3CO3)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.67
ALDH1A1 P00352 3/20 0.67
CYP1A2 P05177 2/20 0.67
KDM4E B2RXH2 1/20 0.67
RAB9A P51151 11/20 0.66
SMN1; SMN2 Q16637 4/20 0.66
TP53 P04637 2/20 0.66
ALOX15 P16050 1/20 0.66
LMNA P02545 2/20 0.64
CASP3 P42574 1/20 0.58
SENP7 Q9BQF6 1/20 0.58
PKM P14618 1/20 0.58
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
P4HTM Q9NXG6 1/20 0.54
MAPT P10636 1/20 0.54
NR4A1 P22736 1/20 0.54
MCL1 Q07820 1/20 0.54
MCHR1 Q99705 1/20 0.54
HIF1A Q16665 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10881661 0.90 NPC1 (0.67) NPC1ALDH1A1CYP1A2KDM4ERAB9A
SCHEMBL14063125 0.89 RAB9A (0.63) NPC1ALDH1A1CYP1A2KDM4ERAB9A
SCHEMBL10735257 0.87 NPC1 (0.78) NPC1ALDH1A1KDM4ERAB9ASMN1; SMN2
SCHEMBL14063123 0.83 NPC1 (0.56) NPC1ALDH1A1CYP1A2KDM4ERAB9A
SCHEMBL5144110 0.82 KMT2A (0.59) NPC1ALDH1A1CYP1A2RAB9ASMN1; SMN2
SCHEMBL9537966 0.82 KMT2A (0.59) NPC1ALDH1A1CYP1A2RAB9ASMN1; SMN2
SCHEMBL410250 0.81 PKM (0.76) ALDH1A1CYP1A2SMN1; SMN2TP53LMNA
SCHEMBL6099389 0.81 PKM (0.76) ALDH1A1CYP1A2SMN1; SMN2TP53LMNA
SCHEMBL5994567 0.81 PKM (0.76) ALDH1A1CYP1A2SMN1; SMN2TP53LMNA
SCHEMBL6799157 0.81 RAB9A (1.00) NPC1ALDH1A1CYP1A2KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0100051-B1 NEW DERIVATIVES OF 1-ALKYLAMINE-(4(P-ALKYLOXY-BENZAMIDE)PHENOXY)-2-PROPANOL, HAVING BETA-SYMPATHOLYTIC ACTIVITY, THEIR SALTS, AND PRODUCTION PROCESSES THEREOF A. Menarini S.a.S. (IT) 1986-04-09 EP disclosed
US-4503075-A ADRENERGIC BLOCKING AGENTS A. MENARINI S.A.S. (IT) 1985-03-05 US disclosed