SCHEMBL10885507

SCHEMBL10885507

O=C(F)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.78
PDK1 Q15118 1/20 0.69
GRM4 Q14833 1/20 0.61
TRPV1 Q8NER1 5/20 0.59
NPSR1 Q6W5P4 2/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA7 P43166 1/20 0.59
CA9 Q16790 1/20 0.59
MEN1 O00255 1/20 0.59
HTT P42858 1/20 0.59
KMT2A Q03164 1/20 0.59
TMPRSS4 Q9NRS4 1/20 0.59
KCNJ5 P48544 1/20 0.59
KCNJ3 P48549 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.58
LMNA P02545 2/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL118026 0.88 KDR (1.00) KDRPDK1GRM4TRPV1CA1
SCHEMBL29364392 0.88 KDR (1.00) KDRPDK1GRM4TRPV1CA1
SCHEMBL9835641 0.86 KDR (0.78) KDRPDK1GRM4TRPV1NPSR1
SCHEMBL11787916 0.86 KDR (0.58) KDRPDK1GRM4TRPV1NPSR1
SCHEMBL2329430 0.86 KDR (0.78) KDRPDK1GRM4TRPV1NPSR1
SCHEMBL31495074 0.85 KDR (0.76) KDRPDK1GRM4TRPV1NPSR1
Fluoride SCHEMBL11788392 0.85 KDR (0.76) KDRPDK1GRM4TRPV1NPSR1
SCHEMBL29759440 0.85 KDR (0.76) KDRPDK1GRM4TRPV1NPSR1
SCHEMBL2457115 0.85 KDR (0.76) KDRPDK1GRM4TRPV1NPSR1
SCHEMBL462753 0.85 KDR (0.76) KDRPDK1GRM4TRPV1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129214-B1 METHOD FOR THE PREPARATION OF BENZENAMINES OCCIDENTAL CHEMICAL CORPORATION (US) 1986-10-29 EP claimed
EP-0129214-A1 Method for the preparation of benzenamines OCCIDENTAL CHEMICAL CORPORATION (US) 1984-12-27 EP claimed
US-4481370-A REACTING HYDROGEN FLUORIDE WITH A PHENYL CARBAMIC FLUORIDE OCCIDENTAL CHEMICAL CORPORATION (US) 1984-11-06 US claimed
EP-0129214-B1 METHOD FOR THE PREPARATION OF BENZENAMINES OCCIDENTAL CHEMICAL CORPORATION (US) 1986-10-29 EP disclosed
US-4481370-A REACTING HYDROGEN FLUORIDE WITH A PHENYL CARBAMIC FLUORIDE OCCIDENTAL CHEMICAL CORPORATION (US) 1984-11-06 US disclosed
US-3983172-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DT) 1976-09-28 US disclosed