SCHEMBL10898516

SCHEMBL10898516

CCCc1ccc(OCCN(CC)CC)cc1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.66
LTA4H P09960 1/20 0.66
CYP2D6 P10635 1/20 0.66
CYP2C9 P11712 1/20 0.66
CYP2C19 P33261 1/20 0.66
HTT P42858 1/20 0.66
KCNH2 Q12809 1/20 0.58
EBP Q15125 1/20 0.58
SIGMAR1 Q99720 1/20 0.58
HRH3 Q9Y5N1 2/20 0.57
MCHR1 Q99705 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18837482 0.91 HRH3 (0.58) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL873540 0.90 CYP1A2 (0.62) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL9706125 0.87 EBP (0.72) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL3973648 0.86 CYP1A2 (0.62) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL8432273 0.85 CYP1A2 (0.70) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL10503798 0.85 CYP2D6 (0.79) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL4547156 0.84 HRH3 (0.79) LTA4HKCNH2HRH3
SCHEMBL873480 0.82 CYP1A2 (0.57) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL9935084 0.82 CYP2D6 (0.66) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19
SCHEMBL6932789 0.82 CYP2D6 (0.66) CYP1A2LTA4HCYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7300936-B2 α-(N-sulfonamido)acetamide derivatives as β-amyloid inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-27 US disclosed
EP-0070133-B1 SECONDARY PHENYLETHANOL AMINES, PROCESSES FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL APPLICATION BEECHAM GROUP PLC (GB) 1986-05-14 EP disclosed