SCHEMBL10909451

SCHEMBL10909451

Cc1ccc(NC(=O)C(=O)Nc2ccc(C)c(C(=O)Nc3ccc4c(O)ccc(S(=O)(=O)O)c4c3)c2)cc1C(=O)Nc1ccc2c(O)ccc(S(=O)(=O)O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNNI3 P19429 1/20 0.46
TNNT2 P45379 1/20 0.46
TNNC1 P63316 1/20 0.46
HKDC1 Q2TB90 1/20 0.46
BRAF P15056 3/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
AKR1C3 P42330 2/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 3/20 0.38
LMNA P02545 2/20 0.38
LDLR P01130 1/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 1/20 0.38
CYP1A2 P05177 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11349822 0.93 TNNI3 (0.46) TNNI3TNNT2TNNC1HKDC1BRAF
SCHEMBL10907979 0.87 BRAF (0.42) BRAFNPC1RAB9ACA12CA1
SCHEMBL10905522 0.85 ENPP2 (0.42) BRAFNPC1RAB9ACA12CA1
SCHEMBL10905262 0.84 BRAF (0.40) TNNI3TNNT2TNNC1HKDC1BRAF
SCHEMBL10908534 0.84 MAOB (0.40) NPC1RAB9AALDH1A1LMNALDLR
SCHEMBL10907419 0.83 BRAF (0.40) TNNI3TNNT2TNNC1HKDC1BRAF
SCHEMBL10907741 0.83 MEN1 (0.45) BRAFALDH1A1LMNAPOLBMAPT
SCHEMBL10907776 0.83 TIMP3 (0.50) TNNI3TNNT2TNNC1HKDC1CA12
SCHEMBL10905258 0.82 TIMP3 (0.44) TNNI3TNNT2TNNC1HKDC1BRAF
SCHEMBL10908593 0.82 NPC1 (0.43) BRAFNPC1RAB9ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4599204-A Oxalylamides useful as dental antiplaque agents and inhibitors of connective tissue destruction AMERICAN CYANAMID COMPANY (US) 1986-07-08 US disclosed