SCHEMBL10915580

SCHEMBL10915580

CC(C)(C#N)Cc1ccc(-c2ccc(CC(C)(C)C#N)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.44
ESR2 Q92731 3/20 0.44
KIF11 P52732 1/20 0.42
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HRH3 Q9Y5N1 6/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP1B1 Q16678 1/20 0.34
SLC6A2 P23975 2/20 0.34
HTR2A P28223 1/20 0.34
SLC6A4 P31645 1/20 0.34
HRH1 P35367 1/20 0.34
HTR2B P41595 1/20 0.34
CHRNA4 P43681 1/20 0.34
SLC6A3 Q01959 1/20 0.34
RXRA P19793 2/20 0.34
RXRB P28702 2/20 0.34
RXRG P48443 2/20 0.34
THRA P10827 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10916780 0.93 ESR1 (0.48) ESR1ESR2KIF11CYP1A1CYP1A2
SCHEMBL2439497 0.84 ESR1 (0.52) ESR1ESR2KIF11TSHRHSD17B10
SCHEMBL971292 0.84 CYP2A6 (0.50) ESR1ESR2TSHRHSD17B10CYP1A1
SCHEMBL2439798 0.84 ESR1 (0.43) ESR1ESR2TSHRCYP1A1CYP1A2
SCHEMBL3160096 0.83 ESR1 (0.42) ESR1ESR2TAAR1
SCHEMBL2823833 0.83 SLC6A4 (0.55) ESR1ESR2CYP1A2SLC6A2HTR2A
SCHEMBL5784144 0.82 SLC6A2 (0.52) ESR1ESR2CYP1A1CYP1A2CYP1B1
SCHEMBL14268192 0.79 ALDH1A1 (0.42) ESR1ESR2TSHRCYP1A1CYP1A2
SCHEMBL27574461 0.78 FDPS (0.40) ESR1ESR2KIF11HSD17B10CYP1A2
SCHEMBL10914831 0.78 HRH3 (0.38) ESR1ESR2HRH3CYP1A2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4564705-A POLYAMIDE, POLYUREA AND POLYURETHANE MONOMERS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-01-14 US disclosed
US-4451642-A Bis(aminoneopentyl) aromatics and polyamides derived therefrom E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-05-29 US disclosed
US-4130579-A Bis(2-methyl-2-cyanopropyl) aromatics E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-12-19 US disclosed