SCHEMBL10918331

SCHEMBL10918331

CC(=O)OC1NC(=O)NC(=O)C1(F)C(=O)OCC(C)C

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.37
ADORA2B P29275 4/20 0.34
ADORA1 P30542 1/20 0.34
MCL1 Q07820 1/20 0.34
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10918279 0.85 ALDH1A1 (0.38) MAPTTSHR
SCHEMBL11245438 0.83 TP53 (0.34)
SCHEMBL11240537 0.80 HSD17B10 (0.39) TSHR
SCHEMBL11235283 0.80 ALDH1A1 (0.39) MAPTADORA2BADORA1MCL1
SCHEMBL11253207 0.76 RGS12 (0.30) TSHR
SCHEMBL11247825 0.74 ALDH1A1 (0.38) MAPTTSHR
SCHEMBL9622596 0.72 ADORA2B (0.42) MAPTADORA2BADORA1
SCHEMBL9622594 0.72 ADORA2B (0.42) MAPTADORA2BADORA1
SCHEMBL11236134 0.71 ALDH1A1 (0.43) MAPTADORA2BTSHR
SCHEMBL11250408 0.71 ALDH1A1 (0.40) MAPTADORA2BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0099091-B1 HEXAHYDRODIOXOPYRIMIDINES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1986-10-29 EP disclosed
US-4536504-A ANTITUMOR, ANTIVIRAL, AND ANTIBACTERIAL AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1985-08-20 US disclosed
EP-0099091-A1 Hexahydrodioxopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1984-01-25 EP disclosed