SCHEMBL10923799

SCHEMBL10923799

COC(=O)Oc1c(C)nc(C)c(OC(=O)OC(C)C)c1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
NPSR1 Q6W5P4 3/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 2/20 0.43
GAA P10253 2/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
RAB9A P51151 1/20 0.43
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
TP53 P04637 1/20 0.39
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
PLA2G2A P14555 1/20 0.38
CACNB4 O00305 1/20 0.38
CACNA1A O00555 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10921719 0.96 SMN1; SMN2 (0.46) SMN1; SMN2NPSR1MAPTKDM4EHPGD
SCHEMBL6955861 0.91 ALDH1A1 (0.49) SMN1; SMN2NPSR1MAPTKDM4EHPGD
SCHEMBL10921995 0.85 SMN1; SMN2 (0.43) SMN1; SMN2NPSR1MAPTKDM4EHPGD
SCHEMBL6962713 0.80 SMN1; SMN2 (0.41) SMN1; SMN2NPSR1MAPTKDM4EHPGD
SCHEMBL6955568 0.77 NPC1 (0.48) SMN1; SMN2NPSR1MAPTKDM4ELMNA
SCHEMBL10920420 0.76 ALDH1A1 (0.46) MAPTHPGDALDH1A1RAB9ACACNB4
SCHEMBL10924017 0.75 AKR1C3 (0.45) SMN1; SMN2MAPTHPGDALDH1A1RAB9A
SCHEMBL11013037 0.75 SMN1; SMN2 (0.63) SMN1; SMN2NPSR1MAPTKDM4EHPGD
SCHEMBL10914513 0.75 DPP4 (0.34) SMN1; SMN2NPSR1MAPTKDM4EHPGD
SCHEMBL11010179 0.74 SMN1; SMN2 (0.66) SMN1; SMN2NPSR1MAPTKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0088938-B1 USE OF PYRIDINE COMPOUNDS FOR THE MANUFACTURE OF MEDICAMENTS WITH AN ANTIHYPOXEMIA AND ISCHEMIA-PROTECTIVE ACTIVITY BAYER AG (DE) 1986-04-30 EP disclosed
EP-0088938-A1 Use of pyridine compounds for the manufacture of medicaments with an antihypoxemia and ischemia-protective activity BAYER AG (DE) 1983-09-21 EP disclosed