SCHEMBL10938263

SCHEMBL10938263

CC(C)N(CCC(C#N)(Cc1ccccc1)C(=O)O)C(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
ALOX15 P16050 2/20 0.42
TSHR P16473 2/20 0.42
SLC22A2 O15244 1/20 0.42
SLC22A1 O15245 1/20 0.42
PGR P06401 1/20 0.42
THRB P10828 1/20 0.42
ADRB3 P13945 1/20 0.42
OPRK1 P41145 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
KCNH2 Q12809 1/20 0.42
PDE3A Q14432 1/20 0.42
SLC47A1 Q96FL8 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
HIF1A Q16665 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9554357 0.79 SMN1; SMN2 (0.52) CYP3A4HIF1ASMN1; SMN2ALDH1A1CYP2C19
SCHEMBL5051285 0.74 SMN1; SMN2 (0.41) CYP3A4HIF1ASMN1; SMN2ALDH1A1CYP2C19
SCHEMBL10942034 0.71 NPC1 (0.36) CYP3A4ALOX15TSHRSLC22A2SLC22A1
SCHEMBL10938259 0.70 CYP3A4 (0.47) CYP3A4ALOX15TSHRSLC22A2SLC22A1
SCHEMBL27515246 0.70 SMN1; SMN2 (0.48) CYP3A4TSHRHIF1ASMN1; SMN2KMT2A
SCHEMBL9555278 0.69 PTPN1 (0.47) CYP3A4TSHRHIF1ASMN1; SMN2MEN1
SCHEMBL6576298 0.69 KCNH2 (0.61) CYP3A4ALOX15TSHRSLC22A2SLC22A1
SCHEMBL11532046 0.69 CYP2D6 (0.46) CYP3A4ALOX15TSHRSLC22A2SLC22A1
SCHEMBL11599547 0.69 CYP2D6 (0.68) CYP3A4ALOX15TSHRSLC22A2SLC22A1
SCHEMBL28561877 0.68 SMN1; SMN2 (0.43) CYP3A4ALOX15TDP1HIF1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4554353-A 2,5-Pyrrolidinedione derivatives useful as antiarrhythmic agents G. D. SEARLE & CO. (US) 1985-11-19 US disclosed