SCHEMBL11599547

SCHEMBL11599547

CC(C)N(CCC(C#N)(c1ccccc1)c1ccccc1)C(C)C

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.68
DRD2 P14416 2/20 0.68
DRD4 P21917 2/20 0.68
OPRM1 P35372 2/20 0.68
DRD3 P35462 2/20 0.68
KCNA3 P22001 7/20 0.48
RAB9A P51151 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CYP3A4 P08684 3/20 0.46
CYP2C19 P33261 1/20 0.46
SLC22A2 O15244 1/20 0.45
SLC22A1 O15245 1/20 0.45
PGR P06401 1/20 0.45
THRB P10828 1/20 0.45
ADRB3 P13945 1/20 0.45
OPRK1 P41145 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
KCNH2 Q12809 1/20 0.45
PDE3A Q14432 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9581143 0.85 CYP3A4 (0.60) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11532046 0.83 CYP2D6 (0.46) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11644267 0.82 CYP2D6 (0.45) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL24683553 0.81 OPRM1 (1.00) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11537087 0.78 EBP (0.50) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11530730 0.78 CYP2D6 (0.56) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL10653133 0.78 CYP3A4 (0.53) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL6258542 0.78 DRD2 (0.68) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11473076 0.77 CYP2D6 (0.46) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11532266 0.76 SIGMAR1 (0.43) CYP2D6DRD2DRD4OPRM1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE29556-E 1,1-Diaryl-1-oxadiazol-alkylamines G. D. SEARLE & CO. (US) 1978-02-28 US disclosed
US-4017491-A 1,1-Diaryl-1H-tetrazole amines G. D. SEARLE & CO. (US) 1977-04-12 US disclosed