SCHEMBL10944802

SCHEMBL10944802

COc1cc(Cc2ncc[nH]2)ccc1OCC(N)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 1/20 0.47
SNCA P37840 1/20 0.46
POLB P06746 3/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
HTT P42858 1/20 0.45
CA2 P00918 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
CREBBP Q92793 1/20 0.42
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10943987 0.86 ALDH1A1 (0.53) ALDH1A1KMT2ACYP2C19CYP1A2MAPT
SCHEMBL11009653 0.79 PPARG (0.49) ALDH1A1POLBHTTKDM4EHPGD
SCHEMBL11008803 0.79 MRGPRX4 (0.48) ALDH1A1CYP2D6CYP2C19CYP1A2POLB
SCHEMBL10945831 0.78 TAAR1 (0.51) ALDH1A1L3MBTL1MEN1KMT2AMAPT
SCHEMBL11009540 0.78 ALDH1A1 (0.45) ALDH1A1CYP2D6CYP2C19CYP1A2MAPT
SCHEMBL19002645 0.76 MEN1 (0.66) ALDH1A1L3MBTL1MEN1KMT2ACYP2D6
SCHEMBL10942106 0.76 MAPT (0.46) ALDH1A1MEN1KMT2ACYP1A2MAPT
SCHEMBL11291865 0.75 CYP19A1 (0.51) ALDH1A1CYP2D6CYP1A2POLBCYP3A4
SCHEMBL12180472 0.73 ACHE (0.60) ALDH1A1L3MBTL1MEN1KMT2ACYP2D6
SCHEMBL11703451 0.73 GAA (0.55) ALDH1A1L3MBTL1MEN1KMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4555516-A FOR TREATMENT OF CARDIOVASCULAR DISORDERS PFIZER INC. (US) 1985-11-26 US disclosed
US-4448781-A CARDIOVASCULAR DISORDERS PFIZER INC. (US) 1984-05-15 US disclosed