SCHEMBL1095000

SCHEMBL1095000

CCNc1cc(Nc2ccc(OCc3cccc(F)c3)c(Cl)c2)ncn1

nearest known ligand 0.78

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.78
ERBB2 P04626 16/20 0.78
GAK O14976 1/20 0.60
ERBB3 P21860 1/20 0.59
ERBB4 Q15303 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094554 0.86 EGFR (0.81) EGFRERBB2GAKERBB3ERBB4
SCHEMBL691455 0.86 EGFR (0.78) EGFRERBB2GAKERBB3ERBB4
SCHEMBL5528646 0.81 EGFR (0.66) EGFRERBB2GAKERBB3ERBB4
SCHEMBL690989 0.80 EGFR (0.65) EGFRERBB2ERBB4
SCHEMBL691623 0.80 EGFR (0.82) EGFRERBB2ERBB4
SCHEMBL2179448 0.79 EGFR (0.60) EGFRERBB2ERBB3
SCHEMBL2177111 0.78 EGFR (0.70) EGFRERBB2ERBB3
SCHEMBL1105303 0.78 EGFR (0.80) EGFRERBB2GAKERBB3ERBB4
SCHEMBL5005468 0.78 EGFR (0.80) EGFRERBB2GAKERBB3ERBB4
SCHEMBL9975357 0.78 EGFR (0.65) EGFRERBB2GAKERBB3ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153791-B2 substituted pyrimidine compoundssuch as 4-amino-6-(3-chloro-4-fluoro-phenylamino)-pyrimidine-5-carbaldehyde O-methyl oxime, used for treating, preventing or ameliorating a chronic or acute protein kinase mediated diseasea, disorders or conditions JANSSEN PHARMACEUTICA N.V. (BE) 2012-04-10 US disclosed