SCHEMBL10955136

SCHEMBL10955136

O=Cc1ccc(Cc2cccnc2)cc1O

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 14/20 0.51
ERN1 O75460 1/20 0.48
MEN1 O00255 1/20 0.45
TP53 P04637 1/20 0.45
CYP3A4 P08684 1/20 0.45
BLM P54132 1/20 0.45
KMT2A Q03164 1/20 0.45
ERCC1 P07992 1/20 0.45
ERCC4 Q92889 1/20 0.45
IDH1 O75874 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10955455 0.88 ERN1 (0.48) TBXAS1ERN1ERCC1ERCC4
SCHEMBL6166029 0.88 ERN1 (0.58) TBXAS1ERN1
SCHEMBL1134433 0.82 IDH1 (0.63) IDH1
SCHEMBL21001943 0.82 CA1 (0.54) MEN1KMT2AIDH1
SCHEMBL10702687 0.81 IDH1 (0.61) TBXAS1MEN1TP53CYP3A4BLM
SCHEMBL8131362 0.79 POLB (0.58) ERN1
SCHEMBL21001935 0.78 IDH1 (0.49) CYP3A4IDH1
SCHEMBL10957763 0.78 TBXAS1 (0.44) TBXAS1ERN1
SCHEMBL10331741 0.77 CA1 (0.65) BLMIDH1
SCHEMBL10331745 0.77 ESR1 (0.54) MEN1KMT2AIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4495357-A THROMBOXANE A2 SYNTHETASE INHIBITORS THE UPJOHN COMPANY (US) 1985-01-22 US disclosed
EP-0069521-A2 Pyridinyl and imidazolyl derivatives of benzofurans and benzothiophenes THE UPJOHN COMPANY (US) 1983-01-12 EP disclosed