SCHEMBL1096396

SCHEMBL1096396

CC(C)(C)C[C@H](c1cccc2ccccc12)N(CC1CCN(c2c(F)cc(C#N)cc2F)CC1c1ccccc1)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
CCR5 P51681 7/20 0.32
DRD3 P35462 1/20 0.32
KCNH2 Q12809 1/20 0.32
CASR P41180 8/20 0.32
CHRM2 P08172 1/20 0.31
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094614 0.94 ESR1 (0.33) ESR1ESR2CCR5DRD3KCNH2
SCHEMBL3575203 0.90 CASR (0.35) CCR5DRD3KCNH2CASR
SCHEMBL1096395 0.85 ESR1 (0.34) ESR1ESR2CCR5DRD3KCNH2
SCHEMBL1096414 0.84 FFAR4 (0.32) CCR5RORC
SCHEMBL3572894 0.84 CASR (0.35) ESR1ESR2CASR
SCHEMBL1096146 0.83 KCNH2 (0.32) CCR5KCNH2
SCHEMBL1094613 0.79 ESR1 (0.34) ESR1ESR2CCR5DRD3KCNH2
SCHEMBL1094794 0.79 FFAR4 (0.32) CCR5
SCHEMBL3573546 0.77 CASR (0.39) CASR
SCHEMBL1096778 0.77 CCR5 (0.39) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153658-B2 Piperidine derivative or salt thereof ASTELLAS PHARMA, INC. (JP) 2012-04-10 US disclosed