SCHEMBL1096778

SCHEMBL1096778

CC(C)(C)C[C@H](c1cccc2ccccc12)N(CC1CCN(C(N)=S)CC1c1cccc(F)c1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.39
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576540 0.89 CCR5 (0.39) CCR5KCNH2
SCHEMBL1096776 0.84 CCR5 (0.39) CCR5KCNH2
SCHEMBL1097414 0.83 CCR5 (0.37) CCR5KCNH2
SCHEMBL1095976 0.80 CCR5 (0.39) CCR5
SCHEMBL1096396 0.77 ESR1 (0.33) CCR5KCNH2
SCHEMBL16274940 0.75 CCR5 (0.44) CCR5
SCHEMBL1105750 0.74 CCR5 (0.40) CCR5KCNH2
SCHEMBL1097192 0.74 HTR2A (0.37) CCR5
SCHEMBL1095663 0.74 CCR5 (0.40) CCR5KCNH2
SCHEMBL1096039 0.74 DPP4 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153658-B2 Piperidine derivative or salt thereof ASTELLAS PHARMA, INC. (JP) 2012-04-10 US disclosed