SCHEMBL10965883

SCHEMBL10965883

N#Cc1cccc(C2CNC(=O)NN2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.47
DRD3 P35462 8/20 0.47
ABCC9 O60706 3/20 0.43
ABCC8 Q09428 3/20 0.43
KCNJ11 Q14654 3/20 0.43
KCNJ8 Q15842 3/20 0.43
CYP19A1 P11511 1/20 0.37
MAOB P27338 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
ALOX5 P09917 1/20 0.35
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
CASP1 P29466 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16431937 0.71 DRD2 (0.56) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL17696870 0.69 DRD2 (0.53) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL10163875 0.69 ABCC9 (0.49) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL1097348 0.69 DRD2 (0.43) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL14869628 0.68 DRD2 (0.76) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL469719 0.68 DRD2 (0.60) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL22456247 0.68 DRD2 (0.60) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL22225174 0.68 DRD2 (0.49) DRD2DRD3ABCC9ABCC8KCNJ11
SCHEMBL28070344 0.68 DRD2 (0.49) DRD2DRD3ABCC9ABCC8KCNJ11
Hydrochloric Acid SCHEMBL31210148 0.67 DRD2 (0.73) DRD2DRD3ABCC9ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0052442-B1 HETEROCYCLIC COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-09-11 EP disclosed