SCHEMBL10967217

SCHEMBL10967217

CC(N)NCC(O)COc1cccc(Cl)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 11/20 0.54
ADRB3 P13945 7/20 0.54
CASR P41180 3/20 0.54
ADRB1 P08588 8/20 0.51
SIGMAR1 Q99720 4/20 0.51
CYP1A2 P05177 4/20 0.51
CYP2D6 P10635 4/20 0.51
HTR2C P28335 4/20 0.51
SLC6A4 P31645 3/20 0.51
HTR2B P41595 3/20 0.51
NR2E1 Q9Y466 3/20 0.51
ALDH1A1 P00352 3/20 0.51
HTR2A P28223 3/20 0.51
HTR6 P50406 3/20 0.51
HTR1A P08908 3/20 0.51
LMNA P02545 3/20 0.51
TSHR P16473 3/20 0.51
MAPK1 P28482 3/20 0.51
SCN1A P35498 2/20 0.51
SLC10A1 Q14973 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10744064 0.90 ADRB2 (0.56) ADRB2ADRB3ADRB1SIGMAR1CYP1A2
SCHEMBL11225584 0.90 ADRB2 (0.63) ADRB2ADRB3ADRB1SIGMAR1CYP1A2
SCHEMBL10738067 0.80 ADRB2 (0.78) ADRB2ADRB3ADRB1SIGMAR1CYP1A2
SCHEMBL10743558 0.80 CYP1A2 (0.60) ADRB2ADRB3ADRB1SIGMAR1CYP1A2
SCHEMBL10965217 0.80 NR2E1 (0.80) ADRB2ADRB3ADRB1SIGMAR1CYP1A2
SCHEMBL10967219 0.80 ADRB2 (0.53) ADRB2ADRB3CASRADRB1CYP1A2
SCHEMBL772732 0.79 NR2E1 (0.58) ADRB2ADRB3CASRCYP1A2CYP2D6
SCHEMBL10737298 0.78 ADRB2 (0.58) ADRB2ADRB3ADRB1SIGMAR1CYP1A2
SCHEMBL5326478 0.77 ADRB2 (0.54) ADRB2ADRB3CASRADRB1SIGMAR1
SCHEMBL11502408 0.77 CYP1A2 (0.57) ADRB2ADRB3CASRCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0057572-B1 ALKANOLAMINE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-07-31 EP disclosed
US-4399138-A DIURETICS, ADRENERGIC BLOCKING AND HYPOTENSIVE AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-08-16 US disclosed