SCHEMBL10967248

SCHEMBL10967248

COC(OC)/C(N)=C/C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.33
SLC1A2 P43004 1/20 0.33
SLC1A1 P43005 1/20 0.33
HCAR2 Q8TDS4 1/20 0.31
GABRP O00591 2/20 0.30
GABRD O14764 2/20 0.30
GABRA1 P14867 2/20 0.30
GABRB1 P18505 2/20 0.30
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30
GABRA5 P31644 2/20 0.30
GABRA3 P34903 2/20 0.30
GABRA2 P47869 2/20 0.30
GABRB2 P47870 2/20 0.30
GABRA4 P48169 2/20 0.30
GABRE P78334 2/20 0.30
GABRA6 Q16445 2/20 0.30
GABRG1 Q8N1C3 2/20 0.30
GABRG3 Q99928 2/20 0.30
GABRQ Q9UN88 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10967253 1.00 SLC1A3 (0.33) SLC1A3SLC1A2SLC1A1HCAR2GABRP
SCHEMBL6539016 0.79 HCAR2 (0.40) HCAR2
SCHEMBL6539020 0.79 HCAR2 (0.40) HCAR2
SCHEMBL11134387 0.79 HCAR2 (0.40) HCAR2
SCHEMBL16612747 0.73 HCAR2 (0.32) SLC1A3SLC1A2SLC1A1HCAR2
SCHEMBL16612748 0.73 HCAR2 (0.32) SLC1A3SLC1A2SLC1A1HCAR2
SCHEMBL10817869 0.73 NPSR1 (0.47) HCAR2
SCHEMBL10817860 0.73 NPSR1 (0.47) HCAR2
SCHEMBL2647447 0.72
SCHEMBL2647446 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023111799-A1 PYRIDINE-3-CARBOXYLATE COMPOUNDS AS CaV1.2 ACTIVATORS NOVARTIS AG (CH) 2023-06-22 WO disclosed
EP-0063359-B1 1,4-DIHYDROPYRIDINE DERIVATIVES AND PROCESSES FOR PREPARING THE SAME BANYU PHARMACEUTICAL CO., LTD. (JP) 1985-12-11 EP disclosed